Elsulfavirine

Name: Elsulfavirine
Brand: Selleck Chemicals
SKU: S6200
Rating: 5 (1 reviews)

Synonyms: Elpida, VM-1500

Catalog No.S6200 Purity:≥99%

Elsulfavirine (Elpida, VM-1500) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) developed for the treatment and prevention of HIV-1 infection.

Elsulfavirine Chemical Structure

CAS No. 868046-19-9

Purity & Quality Control

≥99

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Biological Activity

Description	Elsulfavirine (Elpida, VM-1500) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) developed for the treatment and prevention of HIV-1 infection.

NCT Number	Recruitment	Conditions	Sponsor/Collaborators	Start Date	Phases
Clinical Trial Information (data from https://clinicaltrials.gov, updated on 2024-05-22)
NCT05204394	Unknown status	HIV-1-infection	Viriom	April 1 2022	Phase 2\|Phase 3
NCT05165550	Completed	HIV-1-infection	Viriom	April 12 2022	Phase 1
NCT05163535	Completed	HIV-1-infection	Viriom	January 19 2021	Phase 1\|Phase 2
NCT05148754	Completed	Covid19\|HIV-1-infection	Viriom	January 23 2021	Phase 1
NCT03730311	Unknown status	HIV Infections	Viriom	May 2019	Phase 1
NCT03706911	Completed	HIV-1-infection	Viriom	January 21 2019	Phase 1

Chemical Information & Solubility

Molecular Weight		Formula
CAS No.	868046-19-9	SDF	--
Storage (From the date of receipt)	3 years -20°C powder	Storage of Stock Solutions Aliquot the stock solutions to avoid repeated freeze-thaw cycles	1 year-80°Cin solvent
Storage (From the date of receipt)	3 years -20°C powder		1 month-20°Cin solvent

In vivo
Batch:

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In vivo Formulation Calculator

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In vivo Formulation Calculator (Clear solution)

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH₂O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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