Active Pharmaceutical Ingredients

Catalog No.	Product Name	Information
S2455	Bethanechol chloride	Bethanechol chloride(Myocholine,Urecholine) is a selective muscarinic receptor agonist without any effect on nicotinic receptors.
S1913	Tropicamide	Tropicamide(Ro 1-7683) is an anticholinergic and a muscarinic receptor subtype M4-preferring antagonist with IC50 of 8.0 nM.
S2121	Licofelone (ML3000)	Licofelone (ML3000, Compound 3e) is a dual inhibitor of COX and 5-lipoxygenase (5-LOX) with IC50 of 0.21 μM and 0.18 μM, respectively. Licofelone induces apoptosis, and decreases the production of proinflammatory leukotrienes and prostaglandins. Licofelone is considered as a treatment for osteoarthritis.
S1988	Propylthiouracil	Propylthiouracil (NSC 6498, NSC 70461) is a thyroperoxidase and 5'-deiodinase inhibitor, used to treat hyperthyroidism.
S1830	Oxfendazole	Oxfendazole (RS-8858,Fenbendazole sulfoxide) is a broad spectrum benzimidazole anthelmintic.
S3001	Clevudine	Clevudine(Levovir,L-FMAU) is an antiviral drug for the treatment of hepatitis B.
S2900	Cobicistat	Cobicistat is a potent and selective inhibitor of CYP3A with IC50 of 30-285 nM.
E2363	Etrasimod(APD334)	Etrasimod(APD334) is a potent, selective and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor with an EC50 value of 1.88 nM in CHO cells.
E0109	Fezolinetant	Fezolinetant (ESN-364) is a potential antagonist of the neurokinin 3 receptor (NK3R). It interrupts pulsatile lh secretion and moderates levels of ovarian hormones throughout the menstrual cycle.
S6938	Opicapone	Opicapone(BIA 9-1067) is a potent inhibitor of catechol-O-methyltransferase (COMT) with ED50 values of 1.4 mg⋅kg⁻¹ in rat erythrocytes. It has the potential to be used in research of Parkinson's disease and motor fluctuations.
S6635	Seladelpar	Seladelpar(MBX-8025) is a potent and selective agonist of peroxisome proliferator–activated receptor-delta (PPAR-δ) with EC50 of 2 nM for human PPAR-δ. MBX-8025 enhances insulin sensitivity, counters dyslipidemia, and reduces hepatic storage of lipotoxic lipids, thereby ameliorating NASH pathology in obese diabetic mice.
S9633	GS-6207	GS-6207 (Lenacapavir) is a HIV-1 capsid inhibitor. It shows anti-HIV activity with an EC50 of 0.1 nM in MT-4 cells.

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