Home Endocrinology & Hormones Estrogen/progestogen Receptor antagonist Imlunestrant For research use only.

Imlunestrant

Synonyms: LY3484356

Imlunestrant(LY3484356) is a potent, orally bioavailable selective estrogen receptor degrader (SERD) that functions as a pure antagonist of estrogen receptor alpha (ERα). It inhibits ER-dependent gene transcription and cell proliferation, resulting in sustained suppression of estrogen-driven growth in ER-positive cells.

Imlunestrant Chemical Structure

Imlunestrant Chemical Structure

CAS No. 2408840-26-4

Purity & Quality Control

Imlunestrant Related Products

Signaling Pathway

Estrogen/progestogen Receptor Signaling Pathways

Estrogen/progestogen Receptor Signaling Pathway

Biological Activity

Description Imlunestrant(LY3484356) is a potent, orally bioavailable selective estrogen receptor degrader (SERD) that functions as a pure antagonist of estrogen receptor alpha (ERα). It inhibits ER-dependent gene transcription and cell proliferation, resulting in sustained suppression of estrogen-driven growth in ER-positive cells.

Chemical Information & Solubility

Molecular Weight 524.51 Formula

C29H24F4N2O3
CAS No. 2408840-26-4 SDF Download Imlunestrant SDF
Storage (From the date of receipt)

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

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