Aripiprazole lauroxil

Synonyms: Aristada

Aripiprazole lauroxil(Aristada) is an extended-release prodrug of aripiprazole designed for intramuscular injection. It acts as a dopamine-serotonin system stabilizer, with a potent partial agonist for dopamine D2 and serotonin 5-HT1A receptors while an antagonist for serotonin 5-HT2A receptors.

Aripiprazole lauroxil Chemical Structure

Aripiprazole lauroxil Chemical Structure

CAS No. 1259305-29-7

Purity & Quality Control

Batch: S570701 Ethanol]7 mg/mL]false]DMSO]6 mg/mL]false]Water]Insoluble]false Purity: 99.72%
99.72

Aripiprazole lauroxil Related Products

Biological Activity

Description Aripiprazole lauroxil(Aristada) is an extended-release prodrug of aripiprazole designed for intramuscular injection. It acts as a dopamine-serotonin system stabilizer, with a potent partial agonist for dopamine D2 and serotonin 5-HT1A receptors while an antagonist for serotonin 5-HT2A receptors.

Chemical Information & Solubility

Molecular Weight 660.72 Formula

C36H51Cl2N3O4

CAS No. 1259305-29-7 SDF Download Aripiprazole lauroxil SDF
Storage (From the date of receipt)

In vitro
Batch:

Ethanol : 7 mg/mL

DMSO : 6 mg/mL ( (9.08 mM) Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Water : Insoluble


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In vivo
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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH2O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

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