Home Neuronal Signaling 5-HT Receptor antagonist Azasetron HCl For research use only.

Azasetron HCl

Synonyms: Y-25130 HCl

Azasetron HCl (Y-25130) is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy.

Azasetron HCl Chemical Structure

Azasetron HCl Chemical Structure

CAS No. 123040-16-4

Purity & Quality Control

Azasetron HCl Related Products

Signaling Pathway

5-HT Receptor Signaling Pathways

5-HT Receptor Signaling Pathway

Biological Activity

Description Azasetron HCl (Y-25130) is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy.
Targets
5-HT3 [1]
0.33 nM

Chemical Information & Solubility

Molecular Weight 386.27 Formula

C17H20ClN3O3.HCl
CAS No. 123040-16-4 SDF Download Azasetron HCl SDF
Smiles CN1C(=O)COC2=C(C=C(C=C21)Cl)C(=O)NC3CN4CCC3CC4.Cl
Storage (From the date of receipt)

In vitro
Batch:

Water : 3 mg/mL

DMSO : Insoluble ( Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Ethanol : Insoluble


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