Home Neuronal Signaling 5-HT Receptor antagonist 4F 4PP oxalate For research use only.

4F 4PP oxalate

4F 4PP oxalate is an antagonist of the serotonin (5-HT) receptor subtype 5-HT2A (Ki = 5.3 nM), which is selective for 5-HT2A receptors over 5-HT1C receptors (Ki = 620 nM). 

4F 4PP oxalate Chemical Structure

4F 4PP oxalate Chemical Structure

CAS No. 144734-36-1

Purity & Quality Control

Batch: E007001 DMSO]11 mg/mL]false]Water]Insoluble]false]Ethanol]Insoluble]false Purity: 98.42%
98.42

4F 4PP oxalate Related Products

Signaling Pathway

5-HT Receptor Signaling Pathways

5-HT Receptor Signaling Pathway

Biological Activity

Description 4F 4PP oxalate is an antagonist of the serotonin (5-HT) receptor subtype 5-HT2A (Ki = 5.3 nM), which is selective for 5-HT2A receptors over 5-HT1C receptors (Ki = 620 nM). 
Targets
5-HT2A [1]
(in 5-HT2 binding studies)		 5-HT1C [1]
(in 5-HT1C binding studies)
5.3 nM(Ki) 620 nM(Ki)

Chemical Information & Solubility

Molecular Weight 429.48 Formula

C22H26FNO.C2H2O4
CAS No. 144734-36-1 SDF --
Smiles OC(=O)C(O)=O.FC1=CC=C(C=C1)C(=O)C2CCN(CCCCC3=CC=CC=C3)CC2
Storage (From the date of receipt) 3 years -20°C powder

In vitro
Batch:

DMSO : 11 mg/mL ( (25.61 mM) Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Water : Insoluble

Ethanol : Insoluble


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In vivo
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