Home Neuronal Signaling AChR agonist DREADD agonist 21 For research use only.

DREADD agonist 21

DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (hM3Dq) with EC50 of 1.7 nM.

DREADD agonist 21 Chemical Structure

DREADD agonist 21 Chemical Structure

CAS No. 56296-18-5

Purity & Quality Control

DREADD agonist 21 Related Products

Signaling Pathway

AChR Signaling Pathways

AChR Signaling Pathway

Biological Activity

Description DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (hM3Dq) with EC50 of 1.7 nM.
Targets
hM3Dq [1]
(Cell-free assay)
1.7 nM(EC50)

Chemical Information & Solubility

Molecular Weight 278.35 Formula

C17H18N4
CAS No. 56296-18-5 SDF --
Smiles C1CN(CCN1)C2=NC3=CC=CC=C3NC4=CC=CC=C42
Storage (From the date of receipt) 3 years -20°C powder

In vitro
Batch:

DMSO : 56 mg/mL ( (201.18 mM) Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Ethanol : 56 mg/mL

Water : Insoluble


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