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SGK

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SGK Products

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Catalog No. Product Name Information Product Use Citations Product Validations
S7209 GSK650394 GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively.
J Clin Invest, 2023, 133(20)e169234
J Leukoc Biol, 2023, qiad025
Reprod Biol Endocrinol, 2023, 21(1):50
S9672 PROTAC SGK3 degrader-1 PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC conjugate of the 308-R SGK inhibitor with the VH032 VHL binding ligand, targeting SGK3 (Serum/Glucocorticoid Regulated Kinase Family Member 3) for degradation.
Front Pharmacol, 2023, 14:1169054
Front Pharmacol, 2023, 14:1169054
S8824 EMD638683 EMD638683 is a highly selective inhibitor of serum- and glucocorticoid-inducible kinase 1 (SGK1) with IC50 of 3 μM. EMD638683 exhibits antihypertensive potency and anti-tumor activity.
S7209 GSK650394 GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively.
J Clin Invest, 2023, 133(20)e169234
J Leukoc Biol, 2023, qiad025
Reprod Biol Endocrinol, 2023, 21(1):50
S9672 PROTAC SGK3 degrader-1 PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC conjugate of the 308-R SGK inhibitor with the VH032 VHL binding ligand, targeting SGK3 (Serum/Glucocorticoid Regulated Kinase Family Member 3) for degradation.
Front Pharmacol, 2023, 14:1169054
Front Pharmacol, 2023, 14:1169054
S8824 EMD638683 EMD638683 is a highly selective inhibitor of serum- and glucocorticoid-inducible kinase 1 (SGK1) with IC50 of 3 μM. EMD638683 exhibits antihypertensive potency and anti-tumor activity.

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Tags: SGK inhibitor|SGK agonist|SGK activator|SGK inducer|SGK antagonist|SGK signaling pathway|SGK assay kit