Home Cell Cycle Haspin Kinase

Haspin Kinase

Haspin Kinase Products

  • All (3)
  • Haspin Kinase Inhibitors (3)
  • New Haspin Kinase Products
Catalog No. Product Name Information Product Use Citations Product Validations
S2198 SGI-1776 free base SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 nM in a cell-free assay, 50- and 10-fold selective versus Pim2 and Pim3, also potent to Flt3 and haspin. SGI-1776 induces apoptosis and autophagy.
Cell Death Dis, 2024, 15(9):644
Mar Drugs, 2024, 22(10)444
Mol Cancer, 2023, 22(1):64
S3406 LDN-192960 LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively.
Colloids Surf B Biointerfaces, 2022, 209(Pt 1):112182
E1132 CHR-6494 CHR-6494 is a potent inhibitor of haspin, with an IC50 of 2 nM, inhibits histone H3T3 phosphorylation, and can be used in the research of cancer.
S2198 SGI-1776 free base SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 nM in a cell-free assay, 50- and 10-fold selective versus Pim2 and Pim3, also potent to Flt3 and haspin. SGI-1776 induces apoptosis and autophagy.
Cell Death Dis, 2024, 15(9):644
Mar Drugs, 2024, 22(10)444
Mol Cancer, 2023, 22(1):64
S3406 LDN-192960 LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively.
Colloids Surf B Biointerfaces, 2022, 209(Pt 1):112182
E1132 CHR-6494 CHR-6494 is a potent inhibitor of haspin, with an IC50 of 2 nM, inhibits histone H3T3 phosphorylation, and can be used in the research of cancer.

Choose Selective Haspin Kinase Inhibitors

Tags: Haspin Kinase inhibitor|Haspin Kinase agonist|Haspin Kinase activator|Haspin Kinase inducer|Haspin Kinase antagonist|Haspin Kinase signaling pathway|Haspin Kinase assay kit