Refametinib (R enantiomer)

Name: Refametinib (R enantiomer)
Brand: Selleck Chemicals
SKU: S7058
Rating: 5 (1 reviews)

Synonyms: BAY 869766 R enantiomer, RDEA119 R enantiomer

Catalog No.S7058 Purity:≥99%

Refametinib R enantiomer is a MEK inhibitor extracted from patent WO2007014011A2, compound 1022, has an EC50 of 2.0-15 nM.

Refametinib (R enantiomer) Chemical Structure

CAS No. 923032-38-6

Purity & Quality Control

≥99

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Biological Activity

Description	Refametinib R enantiomer is a MEK inhibitor extracted from patent WO2007014011A2, compound 1022, has an EC50 of 2.0-15 nM.

Chemical Information & Solubility

Molecular Weight	572.34	Formula
CAS No.	923032-38-6	SDF	--
Storage (From the date of receipt)	3 years-20°Cpowder	Solutions are unstable. Prepare fresh or purchase small, pre-packaged sizes. Repackage upon receipt.

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Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH₂O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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