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Penbutolol Sulfate

Name: Penbutolol Sulfate
Brand: Selleck Chemicals
SKU: S9470
Rating: 5 (1 reviews)

Synonyms: (-)-Terbuclomine

Catalog No.S9470 Purity:99.94%

Penbutolol sulfate ((-)-Terbuclomine) is an effective beta-adrenergic receptor blocker and diuretic that is used as an antihypertensive agent.

Penbutolol Sulfate Chemical Structure

CAS No. 38363-32-5

Purity & Quality Control

Batch: Purity: 99.94%

99.94

Penbutolol Sulfate Related Products

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Signaling Pathway

Adrenergic Receptor Signaling Pathway

Biological Activity

Description

Penbutolol sulfate ((-)-Terbuclomine) is an effective beta-adrenergic receptor blocker and diuretic that is used as an antihypertensive agent.

Targets

beta-adrenergic receptor ^[1]

References

[1] Rey AM, et al. Postgrad Med. 1991 Apr;89(5):75-81, 84, 89.

Chemical Information & Solubility

Molecular Weight	680.94	Formula	C₁₈H₂₉NO₂.1/2H₂O₄S
CAS No.	38363-32-5	SDF	--
Smiles	CC(C)(C)NCC(O)COC1=C(C=CC=C1)C2CCCC2.CC(C)(C)NCC(O)COC3=C(C=CC=C3)C4CCCC4.O[S](O)(=O)=O
Storage (From the date of receipt)	3 years -20°C powder	Storage of Stock Solutions Aliquot the stock solutions to avoid repeated freeze-thaw cycles	1 year-80°Cin solvent
Storage (From the date of receipt)	3 years -20°C powder		1 month-20°Cin solvent

In vitro
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In vivo
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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH₂O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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