Nelotanserin

Name: Nelotanserin
Brand: Selleck Chemicals
SKU: E7981
Rating: 5 (1 reviews)

Synonyms: APD125

Catalog No.E7981 Purity:≥99%

Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.

Nelotanserin Chemical Structure

CAS No. 839713-36-9

Purity & Quality Control

≥99

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Biological Activity

Description	Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.

Chemical Information & Solubility

Molecular Weight	437.24	Formula
CAS No.	839713-36-9	SDF	--
Storage (From the date of receipt)	3 years-20°Cpowder	Solutions are unstable. Prepare fresh or purchase small, pre-packaged sizes. Repackage upon receipt.

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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