GR 113808

Name: GR 113808
Brand: Selleck Chemicals
SKU: E7802
Rating: 5 (1 reviews)

Synonyms: null

Catalog No.E7802 Purity:≥99%

GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors.

GR 113808 Chemical Structure

CAS No. 144625-51-4

Purity & Quality Control

≥99

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Biological Activity

Description	GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors.

Chemical Information & Solubility

Molecular Weight	393.50	Formula
CAS No.	144625-51-4	SDF	--
Storage (From the date of receipt)	3 years-20°Cpowder	Solutions are unstable. Prepare fresh or purchase small, pre-packaged sizes. Repackage upon receipt.

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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