LY255283 | 99.83%(HPLC) | In Stock

LY255283 is an antagonist of leukotriene B4 (LTB4) receptor (BLT2) that displaces [3H]LTB4 from its binding site on lung membranes with pKi of 7.0.

LY255283 Chemical Structure

CAS: 117690-79-6

Selleck's LY255283 has been cited by 1 publication

Purity & Quality Control

Batch: S295901 DMSO] 72 mg/mL] false] Water] Insoluble] false] Ethanol] Insoluble] false Purity: 99.83%

99.83

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Biological Activity

Description

LY255283 is an antagonist of leukotriene B4 (LTB4) receptor (BLT2) that displaces [3H]LTB4 from its binding site on lung membranes with pKi of 7.0.

Targets

BLT2 ^[1]
(Cell-free assay)

7.0(pKi)

References
[1] S A Silbaugh, et al. Eur J Pharmacol. 1992 Nov 13;223(1):57-64.

References

[1] S A Silbaugh, et al. Eur J Pharmacol. 1992 Nov 13;223(1):57-64.

Chemical Information & Solubility

Molecular Weight	360.45	Formula	C₁₉H₂₈N₄O₃
CAS No.	117690-79-6	SDF	--
Smiles	CCC1=CC(=C(O)C=C1OCCCCCC(C)(C)C2=N[NH]N=N2)C(C)=O
Storage (From the date of receipt)	3 years -20°C powder	Storage of Stock Solutions Aliquot the stock solutions to avoid repeated freeze-thaw cycles	1 year-80°Cin solvent
Storage (From the date of receipt)	3 years -20°C powder		1 month-20°Cin solvent

In vitro
Batch:

DMSO : 72 mg/mL ( (199.75 mM)； Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Water : Insoluble

Ethanol : Insoluble

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In vivo
Batch:

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Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

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